Journal Articles
151) Dawson J. Konowalchuk, Dennis G. Hall. Divergent Synthesis of 1,2,3,4-Tetrasubstituted Cyclobutenes from a Common Scaffold: Enantioselective Desymmetrization via Dual-Catalyzed Photoredox Cross-Coupling. Angew. Chem. Int. Ed. 2023, 62, e20231350. [Selected as a “Hot Paper” by the Editors]
150) M. Zain H. Kazmi, Olivia M. Schneider, Dennis G. Hall. Expanding the Role of Boron in New Drug Chemotypes: Properties, Chemistry, Pharmaceutical Potential of Hemiboronic Naphthoids. J. Med. Chem. 2023, 66, 13768–13787. [Highlighted in SynFacts]
145) Mohamad Estaitie, Dennis G. Hall. Regiocontrolled Synthesis of Enantioenriched 2-Substituted Dehydropiperidines by Stereospecific Allyl–Allyl Cross-Coupling of a Chiral Allylic Boronate. Chem. Commun. 2022, 58, 1370-1373.
144) Hannah E. Hackney, Dennis G. Hall. Recent Advances in the Luminescence of Arylboronic Acids and their Heteroatom Condensates. ChemPhotoChem. 2022, 6, e202100219.
138) X. Li, D. G. Hall. Synthesis and Applications of β-Aminoalkylboronic Acid Derivatives, Advanced Synthesis & Catalysis 2020, 362, 1-16. [Invited Review article]
136) S. Palvai, J. Bhangu, B. Akgun, C. Moody, D. G. Hall, Y. Brudno. In Vivo Targeting Using Arylboronate/Nopoldiol Click Conjugation, Bioconjugate Chem. 2020, 31, 2288-2292.
133) Y. J. Chen, W. D. Wang, D. Wu, H. B. Zheng, D. G. Hall, R. Narain. Multiresponsive and Self-Healing Hydrogel via Formation of Polymer-Nanogel Interfacial Dynamic Benzoxaborole Esters at Physiological pH, ACS Appl. Mater. Interfaces. 2019, 11, 44742-44750.
132) H. A. Clement, M. Boghi, R. M. McDonald, L. Bernier, J. W. Coe, W. Farrell, C. J. Helal, M. R. Reese, N. W. Sach, J. C. Lee, D. G. Hall. High-Throughput Ligand Screening Enables the Enantioselective Conjugate Borylation of Cyclobutenones to Access Synthetically Versatile Tertiary Cyclobutylboronates, Angew. Chem. Int. Ed. 2019, 58, 18405-18409.
131) M. Paladino, M. Boghi, D. G. Hall. Phenoxy-Dialkoxy Borates as a New Class of Readily Prepared Preactivated Reagents for Base-Free Cross-Coupling, Eur. J. Org. Chem. 2019, 6566-6570.
130) D. G. Hall. Boronic Acid Catalysis, Chem. Soc. Rev. 2019, 48, 3475-3496. [Tutorial Review Article]
129) H.-T. Ang, J. P. G. Rygus, D. G. Hall. Two-component Boronic Acid Catalysis for Increased Reactivity in Challenging Friedel-Crafts Alkylations with Deactivated Benzylic Alcohols, Org. Biomol. Chem. 2019, 17, 6007-6014. [Review Article (refereed)]
128) D. Wu, W. D. Wang, D. Diaz-Dussan, Y. Y. Peng, Y. J. Chen, R. Narain, D. G. Hall. In Situ Forming, Dual-Crosslink Network, Self-Healing Hydrogel Enabled by a Bioorthogonal Nopoldiol-Benzoxaborolate Click Reaction with a Wide pH Range, Chemistry of Materials 2019, 31, 4092-4102.
127) H. A. Clement, D. G. Hall. Synthesis of alpha-Hydroxyalkyl Dehydroazepanes via Catalytic Enantioselective Borylative Migration of an Enol Nonaflate, Tetrahedron Letters 2018, 59, 4334-4339.
126) Y. J. Chen, D. Diaz-Dussan, D. Wu, W. D. Wang, Y. Y. Peng, A. B. Asha, D. G. Hall, K. Ishihara, R. Narain. Bioinspired Self-Healing Hydrogel Based on Benzoxaborole-Catechol Dynamic Covalent Chemistry for 3D Cell Encapsulation, ACS Macro Letters 2018, 7, 904-908.
125) M. Boghi, D. G. Hall. Valdecoxib vs Borazavaldecoxib: Isoxazole B=N Isosterism as a Case Study in Designing and Stabilizing Boron Heterocycles, Org. Biomol. Chem. 2018, 16, 4849-4856.
124) X. Li, D. G. Hall. Diastereocontrolled Protodeboronation of β-Sulfinimido gem-Bis(boronates): A General and Stereoselective Access to α,β-Disubstituted β-Aminoalkylboronates, Angew. Chem. Int. Ed. 2018, 57, 10304-10308.
123) B. Akgun, D. G. Hall. Boronic Acids as Bioorthogonal Probes in Site-Selective Labeling of Proteins, Angew. Chem. Int. Ed. 2018, 57, 13028-13044. [Review Article (refereed)]
122) Z. Shire, M. R. Vakili, T. D. R. Morgan, D. G. Hall, A. Lavasanifar, M. Weinfeld. Nanoencapsulation of Novel Inhibitors of PNKP for Selective Sensitization to Ionizing Radiation and Irinotecan and Induction of Synthetic Lethality, Molecular Pharmaceutics 2018, 15, 2316-2326.
121) X. Mo, T. D. R. Morgan, H. T. Ang, D. G. Hall. Scope and Mechanism of a True Organocatalytic Beckmann Rearrangement with a Boronic Acid / Perfluoropinacol System Under Ambient Conditions, J. Am. Chem. Soc. 2018, 140, 5264-5271.
120) Y. J. Chen, W. D. Wang, D. Wu, M. Nagao, D. G. Hall, T. Thundat, R. Narain. Injectable Self-Healing Zwitterionic Hydrogels Based on Dynamic Benzoxaborole-Sugar Interactions with Tunable Mechanical Properties, Biomacromolecules 2018, 19, 596-605.
119) B. Akgun, C. Li, Y. Hao, G. Lambkin, R. Derda, D. G. Hall. Synergic ‘Click’ Boronate/Thiosemicarbazone System for Fast and Irreversible Bioorthogonal Conjugation in Live Cells, J. Am. Chem. Soc. 2017, 139, 14285-14291.
118) T. Verdelet, R. M. Ward, D. G. Hall. Direct Sulfonamidation of Primary and Secondary Benzylic Alcohols Catalyzed by a Boronic Acid/Oxalic Acid System, Eur. J. Org. Chem. 2017, 5729-5738.
117) D. G. Hall, T. Rybak, T. Verdelet. Multicomponent Hetero-[4 + 2] Cycloaddition/Allylboration Reaction: From Natural Product Synthesis to Drug Discovery, Acc. Chem. Res. 2016, 49, 2489-2500.
116) Y. Wang, L. Li, Y. Kotsuchibashi, S. Vshyvenko, Y. Liu, D. G. Hall, H. Zeng, R. Narain. Injectable Shear-Thinning Hydrogels Based on Dynamic Boronate-Diol Covalent Crosslinking that Spontaneous Self-Healing in Aqueous Media, ACS Biomaterials Sci. & Eng. 2016, 2, 2315-2323.
115) S. Vshyvenko, M. Clapson, I. Suzuki, D. G. Hall. Characterization of the Dynamic Equilibrium Between Close and Open Forms of the Benzoxaborole Pharmacophore. ACS Med. Chem. Lett. 2016, 12, 1097-1101.
114) X. Mo, D. G. Hall. Dual Catalysis Using Boronic Acid and Chiral Amine: Acyclic Quaternary Carbons via Enantioselective Alkylation of Branched Aldehydes with Allylic Alcohols, J. Am. Chem. Soc. 2016, 138, 10762-10765.
113) Y. Kim, D. G. Hall. Optimization and Multigram Scalability of a Catalytic Enantioselective Borylative Migration for the Synthesis of Functionalized Chiral Piperidines, Org. Biomol. Chem. 2016, 4739-4748.
112) B. Akgun, D. G. Hall. Fast and Tight Boronate Formation for ‘Click’ Bioorthogonal Conjugation, Angew. Chem. Int. Ed. 2016, 55, 3909-3913.
111) C. Selin, M. S. Stietz, J. E. Blanchard, S. S. Gehrke, S. Bernard, D. G. Hall, E. M. Brown, S. T. Cardona. A Pipeline for Screening Small Molecules with Growth Inhibitory Activity Against Burkholderia cenocepacia, PLOS One 2015, 10, article # UNSP e0128587.
110) T. Rybak, D.G. Hall. Stereoselective and Regiodivergent Allylic Suzuki-Miyaura Cross-Coupling of 2-Ethoxy Dihydropyranyl Boronates: Synthesis and Confirmation of Absolute Stereochemistry of Diospongin B, Org. Lett. 2015, 17 (17), 4156–4159.
109) X. Mo, J. Yakiwchuk, J. Dansereau, J.A. McCubbin, D.G. Hall. Unsymmetrical Diarylmethanes by Ferroceniumboronic Acid Catalyzed Direct Friedel-Crafts Reactions with Deactivated Benzylic Alcohols: Enhanced Reactivity due to Ion-Pairing Effects, J. Am. Chem. Soc. 2015, 137 (30), 9694-9703.
107) S. Fatemi, N. Gernigon, D.G. Hall. A Multigram-Scale Lower E-Factor Procedure for MIBA-Catalyzed Direct Amidation and its Application to the Coupling of alpha and beta Aminoacids, Green Chemistry 2015, 4016-4028.
106) H. Sun, K. Kubota, D.G. Hall. Reaction Optimization, Scalability, and Mechanistic Insight on the Catalytic Enantioselective Desymmetrization of 1,1-Diborylalkanes via Suzuki-Miyaura Cross Coupling, Chemistry European Journal 2015, in press (DOI: 10.1002/chem.201406680, published online April 1, 2015).
105) Y. Kotsuchibashi, M. Ebara, T. Sato, Y. Wang, R. Rajender, D.G. Hall, R. Narain, T. Aoyagi. Spatiotemporal Control of Synergistic Gel Disintegration Consisting of Boroxole- and Glyco-Based Polymers via Photoinduced Proton Transfer. J. Phys. Chem. B 2015, 119, 2323-2329.
104) C. Ricardo, X. Mo, J.A. McCubbin, D.G. Hall. A Surprising Substituent Effect Provides a Superior Boronic Acid Catalyst for Mild and Metal-Free Direct Friedel-Crafts Alkylations and Prenylations of Neutral Arenes, Chemistry European Journal 2015, 21, 4218-4223.
103) J. Ding, T. Rybak D.G. Hall. Synthesis of Chiral Heterocycles Selectivity by Ligand-Controlled Regiodivergent and Enantiospecific Suzuki-Miyaura Cross-Coupling. Nature Communications 2014, 5, 5474-5482.
102) R.M. Al-Zoubi, D.G. Hall. Catalytic Enantioselective Diversity-Oriented Synthesis of a Small Library of Polyhydroxylated Pyrans Inspired from Thiomarinol Antibiotics, Molecular Diversity 2014, 18, 701-719.
101) H. Zheng, D.G. Hall. Boronic Acid Catalysis: an Atom-Economical Platform for Direct Activation and Functionalization of Carboxylic Acids and Alcohols, Aldrichimica Acta 2014, 47, 41-51.
100) I. Baczko, D. Liknes, W. Yang, K.C. Hamming, G. Searle, K. Jaeger, Z. Husti, V. Juhasz, G. Klausz, R. Pap, L. Saghy, A. Varro, V. Dolinsky, S.H. Wang, V. Rauniyar, D. Hall, J.R.B. Dyck, P.E. Light. Characterization of a Novel Multifunctional Resveratrol Derivative for the Treatment of Atrial Fibrillation, British J. Pharmacol. 2014, 171, 92-106.
99) U. Bhakta, E. Sullivan, D.G. Hall. Catalytic Enantioselective Allylboration of Propargylic Aldehydes, Tetrahedron 2013, 70, 678-683.
98) D. Gao, R. Sand, H. Fu, N. Sharmin, W.J. Gallin, D.G Hall, Synthesis of the Non-peptidic Snail Toxin 6-Bromo-2-mercaptotryptamine Dimer (BrMT2), its Lower and Higher Thio Homologs and Their Ability to Modulate Potassium Ion Channels, Bioorg. Med. Chem. Lett. 2013, 23, 5503-5506.
97) Ding, J.; Hall, D.G. Concise Synthesis and Antimalarial Activity of All Four Mefloquine Stereoisomers Using a Highly Enantioselective Catalytic Borylative Alkene Isomerization, Angewandte Chemie International Edition 2013, 52, 8069-8073.
96) Y. Kotsuchibashi; R.V.C. Agustin; J.-Y. Lu; D. G. Hall; R. Narain; Temperature, pH, and Glucose Responsive Gels via Simple Mixing of Boroxole- and Glyco-Based Polymers, ACS Macro Letters 2013, 2, 260-264.
95) Zimmermann, T.J.; Buerger, M.; Tashiro, E.; Kondoh, Y; Martinez, N.E.; Goermer, K.; Rosin-Steiner, S.; Shimizu, T.; Ozaki, S.; Mikoshiba, K.; Watanabe, N.; Hall, D.; Vetter, I.R.; Osada, H; Hedberg, C; Waldmann, H. Boron-Based Inhibitors of Acyl Protein Thioesterases 1 and 2. ChemBioChem2013, 14, 115-122.
94) N. Gernigon; H. Zheng; D.G. Hall; Solid-Supported Ortho-Iodoarylboronic Acid Catalyst for Direct Amidation of Carboxylic Acids, Tetrahedron Letters, 2013, 54, 4475-4478.
93) H. Zheng; M. Lejkowski; D.G. Hall; Mild Boronic Acid Catalyzed Nazarov Cyclization of Divinyl Alcohols in Tandem with Diels-Alder Cycloaddition, Tetrahedron Letters 2013, 54, 91-94.
92) F. Lizzi; G. Veronesi; F. Belluti; C. Bergamini; A. López-Sánchez; M. Kaiser; R. Brun; R. L. Krauth-Siegel; D.G. Hall; L. Rivas; M.L. Bolognesi; Conjugation of Quinones with Natural Polyamines: Toward an Expanded Antitrypanosomatid Profile. Journal of Medicinal Chemistry 2012, 55, 10490–10500.
91) N. Gernigon; R.M. Al-Zoubi; D.G. Hall; Direct Amidation of Carboxylic Acids Catalyzed by Ortho-Iodo Arylboronic Acids: Catalyst Optimization, Scope, and Preliminary Mechanistic Study Supporting a Peculiar Halogen Acceleration Effect. Journal of Organic Chemistry 2012, 77, 8386-8400. [2012 Journal Of Organic Chemistry Outstanding Paper Of The Year Award (American Chemical Society)]
90) J. Ding; J.C.H. Lee; D.G. Hall; Stereoselective Preparation of β-Aryl-β-Boronyl Enoates and Their Copper-Catalyzed Enantioselective Conjugate Reduction, Organic Letters 2012, 14, 4462-4465.
89) D.G. Hall; J.C.H. Lee; J. Ding; Catalytic Enantioselective Transformations of Borylated Substrates: Preparation and Synthetic Applications of Chiral Alkylboronates, Pure and Applied Chemistry 2012, 84, 2263–2277.
88) H. Zheng; G. Sina; N. Shinji; D.G. Hall; Boronic Acid Catalysis as a Mild and Versatile Strategy for Direct Carbo- and Heterocyclizations of Free Allylic Alcohols, Angewandte Chemie International Edition 2012, 51, 6187-6190.
87) L. Zilke; D.G. Hall; Synthetic Studies Towards the Core Tricyclic Ring System of Pradimicin A, European Journal of Organic Chemistry 2012, 22, 4153-4163.
86) S. Schumacher; F. Grüneberger; M. Katterle; C. Hettrich; D. G. Hall; F.W. Scheller; N.G.-Eichelmann; Molecular Imprinting of Fructose Using a Polymerizable Benzoboroxole: Effective Complexation at pH 7.4, Polymer 2011, 12, 2485-2491.
85) J.W. Tomsho, A. Pal, D.G. Hall, S.J. Benkovic; Ring Structure and Aromatic Substituent Effects on the pKa of the Benzoxaborole Pharmacophore, ACS Medicinal Chemistry Letters 2012, 3, 48-52.
84) S. Schumacher, M. Katterle, C. Hettrich, B.- R. Paulke, D.G. Hall, F.W. Scheller, N.G.-Eichelmann; Label-Free Detection of Enhanced Saccharide Binding at pH 7.4 to Nanoparticulate Benzoboroxole Based Receptor Units, Journal of Molecular Recognition 2011, 6, 953-939.
83) J.C.H. Lee, R. McDonald & D.G. Hall; Enantioselective Preparation and Chemoselective Cross-Coupling of 1,1-Diboron Compounds, Nature Chemistry 2011, 3, 894–899. (Highlighted in Synfacts 2012, 8, 89; Syn Form 2012, 3, A22-A25 (“Syn Story“))
82) J. Ding, D.G. Hall; Preparation of Chiral Secondary Boronic Esters via Copper-Catalyzed Enantioselective Conjugate Reduction of β-Boronyl-β-Alkyl α,β-Unsaturated Esters, Tetrahedron 2012, 68, 3428-3434.
81) H. Zheng, M. Lejkowski, D.G. Hall; Mild and Selective Boronic Acid Catalyzed 1,3-Transposition of Allylic Alcohols and Meyer–Schuster Rearrangement of Propargylic Alcohols, Chemical Science 2011, 2, 1305-1310. [Highlighted in Synfacts 2011, 779]
80) J.C.H. Lee, D.G. Hall; Gold-Catalyzed Cycloisomerization Reactions of Boronated Enynes, Tetrahedron Letters 2011, 51(2), 321-324.
79) J.Y. Lu; D.G. Hall; Fragmentation Enables Complexity in the First Total Synthesis of Vinigrol, Angewandte Chemie International Edition 2010, 49(13), 2286-2288. (Highlight)
78) R. Al-Zoubi, D.G. Hall; Mild Silver(I)-Mediated Regioselective Iodination and Bromination of Arylboronic Acids, Organic Letters 2010, 12(11), 2480-2483.
77) H. Zheng, D.G. Hall; Mild and Efficient Boronic Acid Catalysis of Diels-Alder Cycloadditions to 2-Alkynoic Acids, Tetrahedron Letters 2010, 51(27), 3561-3564.
76) H. Zheng, D.G. Hall; Zirconium-Catalyzed Nagata Reaction for the Synthesis of 2-Aryl-1,3,2-Aryldioxaborins via a Mild Three-Component Condensation of Phenols, Aldehydes, and Boronic Acid, Tetrahedron Letters 2010, 51(32), 4256-4259.
75) J.C.H. Lee, D.G. Hall; Chiral Boronate Derivatives via Catalytic Enantioselective Conjugate Addition of Grignard Reagents on 3-Boronyl Unsaturated Esters and Thioesters, J. Am. Chem. Soc. 2010, 132 (16), 5544–5545. [Highlighted in Synfacts 2010, 795]
74) S. Mothana, J.-M. Grassot, D.G. Hall; Multistep Phase-Switch Synthesis Using Liquid-Liquid Partitioning of Boronic Acids as Productive Phase Tags with an Expanded Repertoire of Compatible Reactions, Angew. Chem. Int. Ed. 2010, 49(16), 2883-2887. [Highlighted in C&EN, March 1, 2010]
73) H. Zheng, R. MacDonald, D.G. Hall; Boronic Acid Catalysis for Mild and Selective [3+2] Dipolar Cycloadditions of Unsaturated Carboxylic Acids, Chem. Eur. J. 2010, 16(18), 5454-5460.
72) T.E. Elford, D.G. Hall; Total Synthesis of (+)-Chinensiolide B via Tandem Allylboration/Lactonization, J. Am. Chem. Soc. 2010, 132(5), 1488–1489.
71) A. Pal, M. Bérubé, D.G. Hall; Design, Synthesis, and Screening of a Library of Peptidyl Bis-Boroxoles as Low Molecular Weight Receptors for Complex Oligosaccharides in Water: Identification of a Receptor for the Tumour Marker TF-Antigen, Angew. Chem. Int. Ed. 2010, 49(8), 1492–1495. [Named a VIP – Very Important Paper] [Highlighted in Nature, 2010 464, 169-170]
70) T.G. Elford, D.G. Hall; Advances in the 2-(Alkoxycarbonyl)allylboration of Carbonyl Compounds and Other Direct Methods for the Preparation of alpha-exo-Alkylidene gamma-Lactones, Synthesis 2010, 6, 893-907.
69) U. Sivasubramaniam, D.G. Hall, Stereoselective Preparation of Oxygenated Heterocycles Using Stereocontrolled Tandem Double-Allylation of Carbonyl Compounds with a Boron-Silicon Reagent, Heterocycles 2010, 80, 1449-1456. [Special issue in honor of Prof. Akira Suzuki]
68) G.K. Freschauf, R.S. Mani, T.R. Mereniuk, M. Fanta, C.A. Virgen, G.L. Dianov, J.-M. Grassot, D.G. Hall, M. Weinfeld; Mechanism of Action of an Imido-piperidine Inhibitor of Human Polynucleotide Kinase/Phosphatase, J. Biol. Chem. 2010, 285, 2351-2360.
67) G. Freschauf, F. Karimi-Busheri, A. Ulaczyk-Lesanko, A. Ahrens, J. Koshy, T. Mereniuk, A. Rasouli-Nia, P. Pasarj, C.F. Holmes, F. Rininsland, D.G. Hall, M. Weinfeld;Identification of a Small Molecule Inhibitor of Human Polynucleotide Kinase/Phosphatase, Cancer Research 2009, 69, 7739-7746.
66) M. Penner, V. Rauniyar, L. Kaspar, D.G. Hall, Catalytic Asymmetric Synthesis of Palmerolide A via Organoboron Methodology, J. Am. Chem. Soc. 2009, 131, 14216-14217.
65) S. Lessard, F. Peng, D.G. Hall, Alpha-Hydroxyalkyl Heterocycles via Chiral Allylic Boronates: Pd-Catalyzed Borylation Leading to a Formal Catalytic Enantioselective Isomerization of Allylic Ether and Amine, J. Am. Chem. Soc. 2009, 131, 9612-9613.
64) B.B. Touré, D.G. Hall, Natural Product Synthesis Using Multicomponent Reaction Strategies, Chemical Reviews 2009, 109, 4439-4486.
63) V. Rauniyar, D.G. Hall, Rationally Improved Chiral Brønsted Acid for Catalytic Enantioselective Allylboration of Aldehydes with an Expanded Reagent Scope, J. Org. Chem. 2009, 74, 4236-4241.
62) L. Carosi, D.G. Hall, Chiral Alpha-substituted Allylboronates in a One-Pot Three-Component Asymmetric Allylic Alkylation / Carbonyl Allylation Reaction Sequence: Applications to the Syntheses of (+)-(3R,5R)-3-Hydroxy-5-Decanolide and (–)-Massoialactone, Canadian Journal of Chemistry 2009, 87, 650-661.
61) T.G. Elford, A. Ulaczyk-Lesanko, G. De Pascale, G. Wright, D.G. Hall, Diversity-Oriented Synthesis and Preliminary Biological Screening of Highly Substituted Five-Membered Lactones and Lactams Originating from an Allylboration Reaction of Aldehydes and Imines, Journal of Combinatorial Chemistry 2009, 11, 155-168.
60) B.H. Kim, C.-H. Yin, Q. Guo, E.A. Bach, H. Lee, C. Sandoval, S. Jayabose, A. Ulaczyk-Lesanko, D.G. Hall, G.-H. Baeg, A Small-Molecule Compound Identified Through a Cell-Based Screening Inhibits JAK/STAT Pathway Signaling in Human Cancer Cells, Molecular Cancer Therapeutics 2008, 7, 2672-2680.
59) T.G. Elford, D.G. Hall, Imine Allylation Using 2-Alkoxycarbonyl Allylboronates as an Expedient Three-Component Reaction to Polysubstituted Alpha-Exo-Methylene-Gamma-Lactams, Tetrahedron Letters 2008, 49, 6995-6998.
58) H. Lachance, O. Marion, D.G. Hall, Synthetic Studies Towards the Pyran Core and Amide Side Chain of Psymberin, Tetrahedron Letters 2008, 49, 6061-6064.
57) M. Bérubé, M. Dowlut, D.G. Hall, Benzoboroxoles as Efficient Glycopyranoside-Binding Agents in Physiological Conditions: Structure and Selectivity of Complex Formation, J. Org. Chem. 2008, 73, 6471-6479. [Selected as a “Feature Article” and for the journal Cover Page]
56) V. Rauniyar, H. Zhai, D.G. Hall; Convenient Preparation of Cycloalkenylboronic Acids Pinacol Esters, Synthetic Communications 2008, 38, 3984-3995.
55) V. Rauniyar, H. Zhai, D.G. Hall; Catalytic Enantioselective Allyl- and Crotylboration of Aldehydes with Chiral Diol-SnCl4 Complexes: Optimization, Substrate Scope and Mechanistic Investigation, J. Am. Chem. Soc. 2008, 130, 8481-8490.
54) R. Al-Zoubi, O. Marion, D.G. Hall; Direct and Waste-Free Amidations and Cycloadditions by Organocatalytic Activation of Carboxylic Acids at Room Temperature, Angewandte Chemie Int. Ed. 2008, 47, 2876-2879. [Selected as a “Hot Paper” by the Editors]
53) O. Marion, X. Gao, S. Marcus, D.G. Hall; Synthesis and Preliminary Antibacterial Evaluation of Simplified Thiomarinol Analogues, Bioorganic and Medicinal Chemistry 2008, 17, 1006-1017.
52) D.G. Hall; Preparation of Allylic Boronates and Applications in Stereoselective Catalytic Allylborations, Pure and Applied Chemistry 2008, 80, 913-927.
51) S. Manku, D.G. Hall; Synthesis, Decoding, and Preliminary Screening of a Bead-Supported Library of Triboronic Acid Receptors for Complex Oligosaccharides, Aust. J. Chem. 2007, 60, 824–828.
50) A. Ulaczyk-Lesanko, E. Pelletier, M. Lee, H. Prinz, H. Waldmann, D. G. Hall; Optimization of Three- and Four-Component Reactions for Polysubstituted Piperidines. Application to the Synthesis and Preliminary Biological Screening of a Prototype Library, Journal of Combinatorial Chemistry 2007, 9, 695-703.
49) V. Rauniyar, D.G. Hall; Preparation of a C2-Symmetric Binol-Derived Diol and its Application in the Catalytic Enantioselective and Catalyst-Controlled Diastereoselective Allylboration of Aldehdyes, Synthesis 2007, 21, 3421–3426.
48) L. Carosi, D. G. Hall; Catalytic Enantioselective Preparation of Alpha-Substituted Allylboronates. One-Pot Addition to Functionalized Aldehydes and a Route to Chiral Allylic Trifluoroborate Salts, Angewandte Chemie Int. Ed. 2007, 46, 5913-5915.
47) Dennis G. Hall; Lewis and Brønsted Acid-Catalyzed Allylboration of Carbonyl Compounds: from Discovery to Mechanism and Applications, Synlett 2007, (Invited Account), 11, 1644-1655.
46) F. Peng, D.G. Hall; Preparation of Alpha-Substituted Allylboronates by Chemoselective Iridium-Catalyzed Asymmetric Allylic Alkylation of 1-Propenylboronates,Tetrahedron Letters 2007, 48, 3305-3309.
45) F. Peng, D.G. Hall; Simple, Stable and Versatile Double-Allylation Reagents for the Stereoselective Preparation of Skeletally Diverse Compounds, J. Am. Chem. Soc. 2007, 129, 3070-3071.
44) S. Mothana, S. Vanneste, N. Chahal, D.G. Hall; Phase-Switch Synthesis with Boronic Acids as Productive Tags, Journal of Combinatorial Chemistry 2007, 193-196.
43) T. Elford, S.H. Yu, Y. Arimura, D.G. Hall; Triflic Acid-Catalyzed Additions of 2-Alkoxycarbonyl Allylboronates to Aldehydes. Study of Scope and Mechanistic Investigation of the Reaction Stereochemistry, J. Org. Chem. 2007, 72, 1276-1284.
42) S. Manku, D.G. Hall; Screening of a Combinatorial Library of Synthetic Polyamines Displaying Selectivity in Multiple Ion Pairing Interactions with Model Polyanionic Compounds in Aqueous Solutions; Journal of Combinatorial Chemistry 2006, 8, 551-561.
41) M. Dowlut, D.G. Hall; An Improved Class of Sugar-Binding Boronic Acids, Soluble and Conjugatable and Capable of Complexing Glycosides in Neutral Water; J. Am. Chem. Soc. 2006, 128, 4226-4227.
40) V. Rauniyar, D.G. Hall; Catalytic Enantioselective and Catalyst-Controlled Diastereofacial-Selective Additions of Allyl- and Crotylboronates to Aldehydes Using Chiral Brønsted Acids. Angewandte Chemie Int. Ed. 2006, 45, 2426-2428.
39) X. Gao, D.G. Hall, M. Deligny, A. Favre, F. Carreaux, B. Carboni; Catalytic Enantioselective Three-Component Hetero-[4+2]Cycloaddition/Allylboration Approach to alpha-Hydroxyalkyl Pyrans: Scope, Limitations, Mechanistic Proposal; Chemistry European Journal 2006, 13, 3132-3142. [Classified a VIP paper]
38) L. Carosi, H. Lachance, D.G. Hall; Additions of Functionalized α-Substituted Allylboronates to Aldehydes Under the Novel Lewis and Brønsted Acid Catalyzed Manifolds,Tetrahedron Letters 2005, 46, 8981-8985.
37) M. Dowlut, O. Hindsgaul, D.G. Hall; Investigation of Non-Specific Effects of Different Dyes in the Screening of Labeled Carbohydrates Against Immobilized Proteins;J. Org. Chem. 2005, 70, 9809-9813.
36) S. H. Yu, M. J. Ferguson, R. McDonald, D. G. Hall; Brønsted Acid-Catalyzed Allylboration: Short and Stereodivergent Synthesis of All Four Eupomatilone Diastereomers with Crystallographic Assignments, J. Am. Chem. Soc. 2005, 127, 12808-12809.
35) D. Li, D.G. Hall; Design and Solid-Phase Synthesis of Chiral Acyclic and Cyclic Diamine Ligands, Tetrahedron Asymmetry 2005, 1733-1736.
34) A. Ulaczyk-Lesanko, D.G. Hall; Wanted: New Multicomponent Reactions for Generating Libraries of Polycyclic Natural Product-Like Compounds, Current Opinion in Chemical Biology 2005, 266-276. [Invited refereed review for June issue]
33) H. Lachance, M. St-Onge, D.G. Hall; Practical and Efficient Multi-Gram Preparation of a Camphor Derived Diol for the Enantioselective Lewis Acid Catalyzed Allylboration of Aldehydes, J. Org. Chem. 2005, 70, 4180-4183.
32) X. Gao, D.G. Hall; Catalytic Asymmetric Synthesis of a Potent Thiomarinol Antibiotic, J. Am. Chem. Soc. 2005, 127, 1628-1629.
[See a highlight of this work in C&EN – Feb. 14 2005]
31) M. Gravel, B.B. Touré, D.G. Hall; Practical Procedure for the Preparation of Functionalized (E)-1-Alkenylboronic Acids Including the Unprecedented 1-Alkoxycarbonyl Derivatives, Org. Prep. Proc. Intl. 2004, 36, 573-579.
30) B. Touré, D.G. Hall; Design of a Nonreductive Method for Chemoselective Cleavage of Hydrazines in the Presence of Unsaturations: Application to a Stereoconvergent Three-Component Synthesis of (-)-Methyl Palustramate; J. Org. Chem. 2004, 69, 8429-8436.
29) M. Gravel, H. Lachance, X. Lu, D.G. Hall; Scope and Limitations of the Scandium-Catalyzed Enantioselective Addition of Chiral Allylboronates to Aldehydes; Synthesis 2004, 1290-1302. [Feature Article].
28) J.W.J. Kennedy, D.G. Hall; Lewis Acid Catalysed Allylboration: Discovery, Optimization, and Application to the Formation of Stereogenic Quaternary Carbon Centres; J. Org. Chem. 2004, 69, 4412-4428.
27) V. Rauniyar, D.G. Hall; Lewis Acids Catalyze The Addition of Allylboronates to Aldehydes by Electrophilic Activation of the Dioxaborolane in a Closed Transition Structure; J. Am. Chem. Soc. 2004, 126, 4518-4519.
26) B. B. Touré, D.G. Hall; Three-Component Aza[4+2]/Allylboration/Retro-sulfinyl-ene Sequential Reaction: A New Stereocontrolled Entry to Palustrine Alkaloids and Other 2,6-Disubstituted Piperidines; Angewandte Chemie Int. Ed. 2004, 43, 2001-2004.
25) D. Stones, S. Manku, X. Lu, D.G. Hall; Modular Solid-Phase Synthetic Approach to Optimize Structural and Electronic Properties of Oligoboronic Acid Receptors and Sensors for the Aqueous Recognition of Oligosaccharides; Chemistry: A European Journal 2004, 10, 92-100.
24) J.W.J. Kennedy, D.G. Hall; Recent Advances in the Activation and Stereochemistry of Boron and Silicon Allylation Reagents; Angewandte Chemie Int. Ed. 2003, 42, 4732-4739. [Minireview]
23) H. Lachance, X. Lu, M. Gravel, D.G. Hall; Scandium-Catalyzed Allylboration of Aldehydes as a Practical Method for Highly Diastereo- and Enantioselective Construction of Homoallylic Alcohols; J. Am. Chem. Soc. 2003, 125, 10160-10161.
22) X. Gao, D.G. Hall; 3-Boronoacrolein as an Exceptional Heterodiene in the Highly Enantio- and Diastereoselective Cr(III)-Catalyzed Three-component [4+2]/Allylboration; J. Am. Chem. Soc. 2003, 125, 9308-9309.
21) J.W.J. Kennedy, D.G. Hall; Design of Chiral Boronate-Substituted Acrylamides. Self-Activation and Remote 1,8-Stereoinduction in [4+2] Cycloaddition; J. Organomet. Chem. 2003, 680, 263-270.
20) N. Zhu, D.G. Hall; Effect of Additives on the Stereochemical Integrity and Reactivity of a-Alkoxycarbonyl Alkenylcopper Intermediates. Optimal Conditions for the Synthesis of Isomerically Pure Tetrasubstituted Alkenes; J. Org. Chem. 2003, 67, 6066-6069.
19) S. Manku, Wang, F.; D.G. Hall; Synthesis and HPLC-ESMS Single-bead Decoding of Split-pool Structural Libraries of Polyamines Supported on Polystyrene and Polystyrene-ethylene Glycol Resins; Journal of Combinatorial Chemistry 2003, 5, 379-391.
18) X. Gao, D.G. Hall; New Electronically Enriched Boronobutadienes for the Synthesis of Hydroxylated Cyclohexenes via Tandem [4+2]/Allylboration; Tetrahedron Lett. 2003, 44, 2231-2235.
17) B.B. Touré, H.R. Hoveyda, J. Tailor, A. Ulaczyk Lesanko, D.G. Hall; A Three-Component Reaction for Diversity-Oriented Synthesis of Polysubstituted Piperidines: Solution and Solid-Phase Optimization of the First Tandem Aza[4+2]/Allylboration; Chemistry: A European Journal 2003, 9, 466-474.
[See a highlight of this work in C&EN – Oct. 27 2003]
16) J.W.J. Kennedy, D.G. Hall; Dramatic Rate Enhancement with Preservation of Stereospecificity in the First Metal-Catalyzed Additions of Allylboronates; J. Am. Chem. Soc. 2002, 124, 11586-11587.
15) D.S. Kopac, D.G. Hall; General Solid-Phase Approach to the Synthesis of Chiral Triazacycloalkane Ligands with Stereogenic Backbone Substituents; Journal of Combinatorial Chemistry 2002, 4, 251-254.
14) J.W.J. Kennedy, D.G. Hall; Novel Isomerically Pure Tetrasubstituted Allylboronates. Stereocontrolled Formation of a-Exomethylene g-Lactones as Aldol-Like Adducts with a Chiral Quaternary Carbon Center; J. Am. Chem. Soc. 2002, 124, 898-899.
13) J.W.J. Kennedy, D.G. Hall; Self-Activation and 1,8-Stereoinduction in a Boronate-Substituted Dienophile; Synlett 2002, 477-479.
12) S. Manku, D.G. Hall; Combinatorial Approach to Selective Multivalent Ion-Pairing in Mixed Aqueous-Organic Media Using Bead-Supported Libraries of Unnatural Polyamines; Organic Letters 2002, 4, 31-34.
11) M. Gravel, K.A. Thompson, M. Zak, C. Berube, D.G. Hall; Universal Solid-Phase Approach to the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids; Journal of Organic Chemistry 2002, 67, 3-15. [This article featured the cover page graphics of this issue]
10) H.R. Hoveyda, D.G. Hall; Solid-Phase Synthesis of Cleavable N-Arylmaleimides: Applications in 1,3-Dipolar Cycloaddition and in Thiol Scavenging; Organic Letters 2001,3, 3491-3494.
9) C. Laplante, D.G. Hall; Direct Mono-N-Methylation of Solid-Supported Amino Acids: A Useful Application of the Matteson Rearrangement of a-Aminoalkylboronic Esters;Organic Letters 2001, 3, 1487-1490.
8) S. Manku, F. Wang, D.G. Hall; Survey of Solution- and Solid-Phase Strategies for the Synthesis and Screening of Libraries Based on Natural Product Templates; Journal of Combinatorial Chemistry 2001, 3, 125-150. [Review]
7) S. Manku, C. Laplante, D. Kopac, T. Chan, D.G. Hall; A Mild and General Solid-Phase Method for the Synthesis of Chiral Polyamines. Solution Studies on the Cleavage of Borane-Amine Intermediates from the Reduction of Secondary Amides; Journal of Organic Chemistry 2001, 66, 874-885.
6) K.A. Thompson, D.G. Hall; Resin-to-Resin Petasis Borono-Mannich Reaction Between Dialkylamino Resins and Supported Boronic Acids; Chemical Communications, 2000, 2379-2380.
5) J. Tailor, D.G. Hall; Tandem Aza[4+2]/Allylboration: A Novel Multicomponent Reaction for the Stereocontrolled Synthesis of a-Hydroxyalkyl Piperidine Derivatives;Organic Letters 2000, 2, 3715-3718.
4) F. Wang, S. Manku, D.G. Hall; Solid Phase Syntheses of Polyamine Toxins HO-416b and PhTX-433. Use of an Efficient Polyamide Reduction Strategy That Facilitates Access to Branched Analogues; Organic Letters 2000, 2, 1581-1583.
3) M. Gravel, C. Bérubé, D.G. Hall; Resin-to-Resin Suzuki Coupling of Solid Supported Arylboronic Acids; Journal of Combinatorial Chemistry 2000, 2, 228-231.
2) D.G. Hall, J. Tailor, M. Gravel. N,N-Diethanolaminomethyl Polystyrene: An Efficient Resin to Immobilize Boronic Acids. Angewandte Chemie International Edition 1999, 38, 3064-3067.
1) D.G. Hall, C. Laplante, S. Manku, J. Nagendran. Mild Oxidative Cleavage of Borane-Amine Adducts from Amide Reductions. Efficient Solution- and Solid-Phase Synthesis of N-Alkyl Aminoacids and Chiral Oligoamines. Journal of Organic Chemistry 1999, 64, 698-699.
Other
D.G. Hall; Combinatorial Chemistry Gives Cell Biology Some Muscle Nature Biotechnology 2000, 18, 261-262.
D. Hall; Combinatorial Chemistry – A Powerful Approach to Supermolecule Discovery; Canadian Chemical News, October 1997, 23-25.
78) R. Al-Zoubi, D.G. Hall; Mild Silver(I)-Mediated Regioselective Iodination and Bromination of Arylboronic Acids, Organic Letters 2010, 12(11), 2480-2483.
77) H. Zheng, D.G. Hall; Mild and Efficient Boronic Acid Catalysis of Diels-Alder Cycloadditions to 2-Alkynoic Acids, Tetrahedron Letters 2010, 51(27), 3561-3564.
76) H. Zheng, D.G. Hall; Zirconium-Catalyzed Nagata Reaction for the Synthesis of 2-Aryl-1,3,2-Aryldioxaborins via a Mild Three-Component Condensation of Phenols, Aldehydes, and Boronic Acid, Tetrahedron Letters 2010, 51(32), 4256-4259.
75) J.C.H. Lee, D.G. Hall; Chiral Boronate Derivatives via Catalytic Enantioselective Conjugate Addition of Grignard Reagents on 3-Boronyl Unsaturated Esters and Thioesters, J. Am. Chem. Soc. 2010, 132 (16), 5544–5545. [Highlighted in Synfacts 2010, 795]
74) S. Mothana, J.-M. Grassot, D.G. Hall; Multistep Phase-Switch Synthesis Using Liquid-Liquid Partitioning of Boronic Acids as Productive Phase Tags with an Expanded Repertoire of Compatible Reactions, Angew. Chem. Int. Ed. 2010, 49(16), 2883-2887. [Highlighted in C&EN, March 1, 2010]
73) H. Zheng, R. MacDonald, D.G. Hall; Boronic Acid Catalysis for Mild and Selective [3+2] Dipolar Cycloadditions of Unsaturated Carboxylic Acids, Chem. Eur. J. 2010, 16(18), 5454-5460.
72) T.E. Elford, D.G. Hall; Total Synthesis of (+)-Chinensiolide B via Tandem Allylboration/Lactonization, J. Am. Chem. Soc. 2010, 132(5), 1488–1489.
71) A. Pal, M. Bérubé, D.G. Hall; Design, Synthesis, and Screening of a Library of Peptidyl Bis-Boroxoles as Low Molecular Weight Receptors for Complex Oligosaccharides in Water: Identification of a Receptor for the Tumour Marker TF-Antigen, Angew. Chem. Int. Ed. 2010, 49(8), 1492–1495. [Named a VIP – Very Important Paper] [Highlighted in Nature, 2010 464, 169-170]
70) T.G. Elford, D.G. Hall; Advances in the 2-(Alkoxycarbonyl)allylboration of Carbonyl Compounds and Other Direct Methods for the Preparation of alpha-exo-Alkylidene gamma-Lactones, Synthesis 2010, 6, 893-907.
69) U. Sivasubramaniam, D.G. Hall, Stereoselective Preparation of Oxygenated Heterocycles Using Stereocontrolled Tandem Double-Allylation of Carbonyl Compounds with a Boron-Silicon Reagent, Heterocycles 2010, 80, 1449-1456. [Special issue in honor of Prof. Akira Suzuki]
68) G.K. Freschauf, R.S. Mani, T.R. Mereniuk, M. Fanta, C.A. Virgen, G.L. Dianov, J.-M. Grassot, D.G. Hall, M. Weinfeld; Mechanism of Action of an Imido-piperidine Inhibitor of Human Polynucleotide Kinase/Phosphatase, J. Biol. Chem. 2010, 285, 2351-2360.
67) G. Freschauf, F. Karimi-Busheri, A. Ulaczyk-Lesanko, A. Ahrens, J. Koshy, T. Mereniuk, A. Rasouli-Nia, P. Pasarj, C.F. Holmes, F. Rininsland, D.G. Hall, M. Weinfeld;Identification of a Small Molecule Inhibitor of Human Polynucleotide Kinase/Phosphatase, Cancer Research 2009, 69, 7739-7746.
66) M. Penner, V. Rauniyar, L. Kaspar, D.G. Hall, Catalytic Asymmetric Synthesis of Palmerolide A via Organoboron Methodology, J. Am. Chem. Soc. 2009, 131, 14216-14217.
65) S. Lessard, F. Peng, D.G. Hall, Alpha-Hydroxyalkyl Heterocycles via Chiral Allylic Boronates: Pd-Catalyzed Borylation Leading to a Formal Catalytic Enantioselective Isomerization of Allylic Ether and Amine, J. Am. Chem. Soc. 2009, 131, 9612-9613.
64) B.B. Touré, D.G. Hall, Natural Product Synthesis Using Multicomponent Reaction Strategies, Chemical Reviews 2009, 109, 4439-4486.
63) V. Rauniyar, D.G. Hall, Rationally Improved Chiral Brønsted Acid for Catalytic Enantioselective Allylboration of Aldehydes with an Expanded Reagent Scope, J. Org. Chem. 2009, 74, 4236-4241.
62) L. Carosi, D.G. Hall, Chiral Alpha-substituted Allylboronates in a One-Pot Three-Component Asymmetric Allylic Alkylation / Carbonyl Allylation Reaction Sequence: Applications to the Syntheses of (+)-(3R,5R)-3-Hydroxy-5-Decanolide and (–)-Massoialactone, Canadian Journal of Chemistry 2009, 87, 650-661.
61) T.G. Elford, A. Ulaczyk-Lesanko, G. De Pascale, G. Wright, D.G. Hall, Diversity-Oriented Synthesis and Preliminary Biological Screening of Highly Substituted Five-Membered Lactones and Lactams Originating from an Allylboration Reaction of Aldehydes and Imines, Journal of Combinatorial Chemistry 2009, 11, 155-168.
60) B.H. Kim, C.-H. Yin, Q. Guo, E.A. Bach, H. Lee, C. Sandoval, S. Jayabose, A. Ulaczyk-Lesanko, D.G. Hall, G.-H. Baeg, A Small-Molecule Compound Identified Through a Cell-Based Screening Inhibits JAK/STAT Pathway Signaling in Human Cancer Cells, Molecular Cancer Therapeutics 2008, 7, 2672-2680.
59) T.G. Elford, D.G. Hall, Imine Allylation Using 2-Alkoxycarbonyl Allylboronates as an Expedient Three-Component Reaction to Polysubstituted Alpha-Exo-Methylene-Gamma-Lactams, Tetrahedron Letters 2008, 49, 6995-6998.
58) H. Lachance, O. Marion, D.G. Hall, Synthetic Studies Towards the Pyran Core and Amide Side Chain of Psymberin, Tetrahedron Letters 2008, 49, 6061-6064.
57) M. Bérubé, M. Dowlut, D.G. Hall, Benzoboroxoles as Efficient Glycopyranoside-Binding Agents in Physiological Conditions: Structure and Selectivity of Complex Formation, J. Org. Chem. 2008, 73, 6471-6479. [Selected as a “Feature Article” and for the journal Cover Page]
56) V. Rauniyar, H. Zhai, D.G. Hall; Convenient Preparation of Cycloalkenylboronic Acids Pinacol Esters, Synthetic Communications 2008, 38, 3984-3995.
55) V. Rauniyar, H. Zhai, D.G. Hall; Catalytic Enantioselective Allyl- and Crotylboration of Aldehydes with Chiral Diol-SnCl4 Complexes: Optimization, Substrate Scope and Mechanistic Investigation, J. Am. Chem. Soc. 2008, 130, 8481-8490.
54) R. Al-Zoubi, O. Marion, D.G. Hall; Direct and Waste-Free Amidations and Cycloadditions by Organocatalytic Activation of Carboxylic Acids at Room Temperature, Angewandte Chemie Int. Ed. 2008, 47, 2876-2879. [Selected as a “Hot Paper” by the Editors]
53) O. Marion, X. Gao, S. Marcus, D.G. Hall; Synthesis and Preliminary Antibacterial Evaluation of Simplified Thiomarinol Analogues, Bioorganic and Medicinal Chemistry 2008, 17, 1006-1017.
52) D.G. Hall; Preparation of Allylic Boronates and Applications in Stereoselective Catalytic Allylborations, Pure and Applied Chemistry 2008, 80, 913-927.
51) S. Manku, D.G. Hall; Synthesis, Decoding, and Preliminary Screening of a Bead-Supported Library of Triboronic Acid Receptors for Complex Oligosaccharides, Aust. J. Chem. 2007, 60, 824–828.
50) A. Ulaczyk-Lesanko, E. Pelletier, M. Lee, H. Prinz, H. Waldmann, D. G. Hall; Optimization of Three- and Four-Component Reactions for Polysubstituted Piperidines. Application to the Synthesis and Preliminary Biological Screening of a Prototype Library, Journal of Combinatorial Chemistry 2007, 9, 695-703.
49) V. Rauniyar, D.G. Hall; Preparation of a C2-Symmetric Binol-Derived Diol and its Application in the Catalytic Enantioselective and Catalyst-Controlled Diastereoselective Allylboration of Aldehdyes, Synthesis 2007, 21, 3421–3426.
48) L. Carosi, D. G. Hall; Catalytic Enantioselective Preparation of Alpha-Substituted Allylboronates. One-Pot Addition to Functionalized Aldehydes and a Route to Chiral Allylic Trifluoroborate Salts, Angewandte Chemie Int. Ed. 2007, 46, 5913-5915.
47) Dennis G. Hall; Lewis and Brønsted Acid-Catalyzed Allylboration of Carbonyl Compounds: from Discovery to Mechanism and Applications, Synlett 2007, (Invited Account), 11, 1644-1655.
46) F. Peng, D.G. Hall; Preparation of Alpha-Substituted Allylboronates by Chemoselective Iridium-Catalyzed Asymmetric Allylic Alkylation of 1-Propenylboronates,Tetrahedron Letters 2007, 48, 3305-3309.
45) F. Peng, D.G. Hall; Simple, Stable and Versatile Double-Allylation Reagents for the Stereoselective Preparation of Skeletally Diverse Compounds, J. Am. Chem. Soc. 2007, 129, 3070-3071.
44) S. Mothana, S. Vanneste, N. Chahal, D.G. Hall; Phase-Switch Synthesis with Boronic Acids as Productive Tags, Journal of Combinatorial Chemistry 2007, 193-196.
43) T. Elford, S.H. Yu, Y. Arimura, D.G. Hall; Triflic Acid-Catalyzed Additions of 2-Alkoxycarbonyl Allylboronates to Aldehydes. Study of Scope and Mechanistic Investigation of the Reaction Stereochemistry, J. Org. Chem. 2007, 72, 1276-1284.
42) S. Manku, D.G. Hall; Screening of a Combinatorial Library of Synthetic Polyamines Displaying Selectivity in Multiple Ion Pairing Interactions with Model Polyanionic Compounds in Aqueous Solutions; Journal of Combinatorial Chemistry 2006, 8, 551-561.
41) M. Dowlut, D.G. Hall; An Improved Class of Sugar-Binding Boronic Acids, Soluble and Conjugatable and Capable of Complexing Glycosides in Neutral Water; J. Am. Chem. Soc. 2006, 128, 4226-4227.
40) V. Rauniyar, D.G. Hall; Catalytic Enantioselective and Catalyst-Controlled Diastereofacial-Selective Additions of Allyl- and Crotylboronates to Aldehydes Using Chiral Brønsted Acids. Angewandte Chemie Int. Ed. 2006, 45, 2426-2428.
39) X. Gao, D.G. Hall, M. Deligny, A. Favre, F. Carreaux, B. Carboni; Catalytic Enantioselective Three-Component Hetero-[4+2]Cycloaddition/Allylboration Approach to alpha-Hydroxyalkyl Pyrans: Scope, Limitations, Mechanistic Proposal; Chemistry European Journal 2006, 13, 3132-3142. [Classified a VIP paper]
38) L. Carosi, H. Lachance, D.G. Hall; Additions of Functionalized α-Substituted Allylboronates to Aldehydes Under the Novel Lewis and Brønsted Acid Catalyzed Manifolds,Tetrahedron Letters 2005, 46, 8981-8985.
37) M. Dowlut, O. Hindsgaul, D.G. Hall; Investigation of Non-Specific Effects of Different Dyes in the Screening of Labeled Carbohydrates Against Immobilized Proteins;J. Org. Chem. 2005, 70, 9809-9813.
36) S. H. Yu, M. J. Ferguson, R. McDonald, D. G. Hall; Brønsted Acid-Catalyzed Allylboration: Short and Stereodivergent Synthesis of All Four Eupomatilone Diastereomers with Crystallographic Assignments, J. Am. Chem. Soc. 2005, 127, 12808-12809.
35) D. Li, D.G. Hall; Design and Solid-Phase Synthesis of Chiral Acyclic and Cyclic Diamine Ligands, Tetrahedron Asymmetry 2005, 1733-1736.
34) A. Ulaczyk-Lesanko, D.G. Hall; Wanted: New Multicomponent Reactions for Generating Libraries of Polycyclic Natural Product-Like Compounds, Current Opinion in Chemical Biology 2005, 266-276. [Invited refereed review for June issue]
33) H. Lachance, M. St-Onge, D.G. Hall; Practical and Efficient Multi-Gram Preparation of a Camphor Derived Diol for the Enantioselective Lewis Acid Catalyzed Allylboration of Aldehydes, J. Org. Chem. 2005, 70, 4180-4183.
32) X. Gao, D.G. Hall; Catalytic Asymmetric Synthesis of a Potent Thiomarinol Antibiotic, J. Am. Chem. Soc. 2005, 127, 1628-1629.
[See a highlight of this work in C&EN – Feb. 14 2005]
31) M. Gravel, B.B. Touré, D.G. Hall; Practical Procedure for the Preparation of Functionalized (E)-1-Alkenylboronic Acids Including the Unprecedented 1-Alkoxycarbonyl Derivatives, Org. Prep. Proc. Intl. 2004, 36, 573-579.
30) B. Touré, D.G. Hall; Design of a Nonreductive Method for Chemoselective Cleavage of Hydrazines in the Presence of Unsaturations: Application to a Stereoconvergent Three-Component Synthesis of (-)-Methyl Palustramate; J. Org. Chem. 2004, 69, 8429-8436.
29) M. Gravel, H. Lachance, X. Lu, D.G. Hall; Scope and Limitations of the Scandium-Catalyzed Enantioselective Addition of Chiral Allylboronates to Aldehydes; Synthesis 2004, 1290-1302. [Feature Article].
28) J.W.J. Kennedy, D.G. Hall; Lewis Acid Catalysed Allylboration: Discovery, Optimization, and Application to the Formation of Stereogenic Quaternary Carbon Centres; J. Org. Chem. 2004, 69, 4412-4428.
27) V. Rauniyar, D.G. Hall; Lewis Acids Catalyze The Addition of Allylboronates to Aldehydes by Electrophilic Activation of the Dioxaborolane in a Closed Transition Structure; J. Am. Chem. Soc. 2004, 126, 4518-4519.
26) B. B. Touré, D.G. Hall; Three-Component Aza[4+2]/Allylboration/Retro-sulfinyl-ene Sequential Reaction: A New Stereocontrolled Entry to Palustrine Alkaloids and Other 2,6-Disubstituted Piperidines; Angewandte Chemie Int. Ed. 2004, 43, 2001-2004.
25) D. Stones, S. Manku, X. Lu, D.G. Hall; Modular Solid-Phase Synthetic Approach to Optimize Structural and Electronic Properties of Oligoboronic Acid Receptors and Sensors for the Aqueous Recognition of Oligosaccharides; Chemistry: A European Journal 2004, 10, 92-100.
24) J.W.J. Kennedy, D.G. Hall; Recent Advances in the Activation and Stereochemistry of Boron and Silicon Allylation Reagents; Angewandte Chemie Int. Ed. 2003, 42, 4732-4739. [Minireview]
23) H. Lachance, X. Lu, M. Gravel, D.G. Hall; Scandium-Catalyzed Allylboration of Aldehydes as a Practical Method for Highly Diastereo- and Enantioselective Construction of Homoallylic Alcohols; J. Am. Chem. Soc. 2003, 125, 10160-10161.
22) X. Gao, D.G. Hall; 3-Boronoacrolein as an Exceptional Heterodiene in the Highly Enantio- and Diastereoselective Cr(III)-Catalyzed Three-component [4+2]/Allylboration; J. Am. Chem. Soc. 2003, 125, 9308-9309.
21) J.W.J. Kennedy, D.G. Hall; Design of Chiral Boronate-Substituted Acrylamides. Self-Activation and Remote 1,8-Stereoinduction in [4+2] Cycloaddition; J. Organomet. Chem. 2003, 680, 263-270.
20) N. Zhu, D.G. Hall; Effect of Additives on the Stereochemical Integrity and Reactivity of a-Alkoxycarbonyl Alkenylcopper Intermediates. Optimal Conditions for the Synthesis of Isomerically Pure Tetrasubstituted Alkenes; J. Org. Chem. 2003, 67, 6066-6069.
19) S. Manku, Wang, F.; D.G. Hall; Synthesis and HPLC-ESMS Single-bead Decoding of Split-pool Structural Libraries of Polyamines Supported on Polystyrene and Polystyrene-ethylene Glycol Resins; Journal of Combinatorial Chemistry 2003, 5, 379-391.
18) X. Gao, D.G. Hall; New Electronically Enriched Boronobutadienes for the Synthesis of Hydroxylated Cyclohexenes via Tandem [4+2]/Allylboration; Tetrahedron Lett. 2003, 44, 2231-2235.
17) B.B. Touré, H.R. Hoveyda, J. Tailor, A. Ulaczyk Lesanko, D.G. Hall; A Three-Component Reaction for Diversity-Oriented Synthesis of Polysubstituted Piperidines: Solution and Solid-Phase Optimization of the First Tandem Aza[4+2]/Allylboration; Chemistry: A European Journal 2003, 9, 466-474.
[See a highlight of this work in C&EN – Oct. 27 2003]
16) J.W.J. Kennedy, D.G. Hall; Dramatic Rate Enhancement with Preservation of Stereospecificity in the First Metal-Catalyzed Additions of Allylboronates; J. Am. Chem. Soc. 2002, 124, 11586-11587.
15) D.S. Kopac, D.G. Hall; General Solid-Phase Approach to the Synthesis of Chiral Triazacycloalkane Ligands with Stereogenic Backbone Substituents; Journal of Combinatorial Chemistry 2002, 4, 251-254.
14) J.W.J. Kennedy, D.G. Hall; Novel Isomerically Pure Tetrasubstituted Allylboronates. Stereocontrolled Formation of a-Exomethylene g-Lactones as Aldol-Like Adducts with a Chiral Quaternary Carbon Center; J. Am. Chem. Soc. 2002, 124, 898-899.
13) J.W.J. Kennedy, D.G. Hall; Self-Activation and 1,8-Stereoinduction in a Boronate-Substituted Dienophile; Synlett 2002, 477-479.
12) S. Manku, D.G. Hall; Combinatorial Approach to Selective Multivalent Ion-Pairing in Mixed Aqueous-Organic Media Using Bead-Supported Libraries of Unnatural Polyamines; Organic Letters 2002, 4, 31-34.
11) M. Gravel, K.A. Thompson, M. Zak, C. Berube, D.G. Hall; Universal Solid-Phase Approach to the Immobilization, Derivatization, and Resin-to-Resin Transfer Reactions of Boronic Acids; Journal of Organic Chemistry 2002, 67, 3-15. [This article featured the cover page graphics of this issue]
10) H.R. Hoveyda, D.G. Hall; Solid-Phase Synthesis of Cleavable N-Arylmaleimides: Applications in 1,3-Dipolar Cycloaddition and in Thiol Scavenging; Organic Letters 2001,3, 3491-3494.
9) C. Laplante, D.G. Hall; Direct Mono-N-Methylation of Solid-Supported Amino Acids: A Useful Application of the Matteson Rearrangement of a-Aminoalkylboronic Esters;Organic Letters 2001, 3, 1487-1490.
8) S. Manku, F. Wang, D.G. Hall; Survey of Solution- and Solid-Phase Strategies for the Synthesis and Screening of Libraries Based on Natural Product Templates; Journal of Combinatorial Chemistry 2001, 3, 125-150. [Review]
7) S. Manku, C. Laplante, D. Kopac, T. Chan, D.G. Hall; A Mild and General Solid-Phase Method for the Synthesis of Chiral Polyamines. Solution Studies on the Cleavage of Borane-Amine Intermediates from the Reduction of Secondary Amides; Journal of Organic Chemistry 2001, 66, 874-885.
6) K.A. Thompson, D.G. Hall; Resin-to-Resin Petasis Borono-Mannich Reaction Between Dialkylamino Resins and Supported Boronic Acids; Chemical Communications, 2000, 2379-2380.
5) J. Tailor, D.G. Hall; Tandem Aza[4+2]/Allylboration: A Novel Multicomponent Reaction for the Stereocontrolled Synthesis of a-Hydroxyalkyl Piperidine Derivatives;Organic Letters 2000, 2, 3715-3718.
4) F. Wang, S. Manku, D.G. Hall; Solid Phase Syntheses of Polyamine Toxins HO-416b and PhTX-433. Use of an Efficient Polyamide Reduction Strategy That Facilitates Access to Branched Analogues; Organic Letters 2000, 2, 1581-1583.
3) M. Gravel, C. Bérubé, D.G. Hall; Resin-to-Resin Suzuki Coupling of Solid Supported Arylboronic Acids; Journal of Combinatorial Chemistry 2000, 2, 228-231.
2) D.G. Hall, J. Tailor, M. Gravel. N,N-Diethanolaminomethyl Polystyrene: An Efficient Resin to Immobilize Boronic Acids. Angewandte Chemie International Edition 1999, 38, 3064-3067.
1) D.G. Hall, C. Laplante, S. Manku, J. Nagendran. Mild Oxidative Cleavage of Borane-Amine Adducts from Amide Reductions. Efficient Solution- and Solid-Phase Synthesis of N-Alkyl Aminoacids and Chiral Oligoamines. Journal of Organic Chemistry 1999, 64, 698-699.
Other
D.G. Hall; Combinatorial Chemistry Gives Cell Biology Some Muscle Nature Biotechnology 2000, 18, 261-262.
D. Hall; Combinatorial Chemistry – A Powerful Approach to Supermolecule Discovery; Canadian Chemical News, October 1997, 23-25.
